In this article we will explore the fascinating world of SR-144,528 and its impact on our lives. SR-144,528 has been a fundamental figure in human history, playing a crucial role in various aspects, from science and technology to culture and art. Over the years, SR-144,528 has aroused great interest and has been the subject of study and research, revealing surprising aspects that have revolutionized our view of the world. In this article, we will analyze the different facets of SR-144,528 and its influence on human development, offering a deep and enriching look at this exciting topic.
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Formula | C29H34ClN3O |
Molar mass | 476.06 g·mol−1 |
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SR144528 is a drug that acts as a potent and highly selective CB2 receptor inverse agonist, with a Ki of 0.6 nM at CB2 and 400 nM at the related CB1 receptor. It is used in scientific research for investigating the function of the CB2 receptor, as well as for studying the effects of CB1 receptors in isolation, as few CB1 agonists that do not also show significant activity as CB2 agonists are available. It has also been found to be an inhibitor of sterol O-acyltransferase, an effect that appears to be independent from its action on CB2 receptors.